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OPRM1 and GRM1
Data Source:
BioGRID
(two hybrid)
OPRM1
GRM1
Description
opioid receptor mu 1
glutamate metabotropic receptor 1
Image
No pdb structure
GO Annotations
Cellular Component
Endosome
Endoplasmic Reticulum
Golgi Apparatus
Plasma Membrane
Integral Component Of Plasma Membrane
Focal Adhesion
Axon
Dendrite
Dendrite Membrane
Dendrite Cytoplasm
Sarcolemma
Neuron Projection
Perikaryon
Membrane Raft
Spine Apparatus
Integral Component Of Postsynaptic Membrane
Integral Component Of Presynaptic Membrane
Nucleus
Plasma Membrane
Integral Component Of Plasma Membrane
Dendrite
G Protein-coupled Receptor Dimeric Complex
G Protein-coupled Receptor Homodimeric Complex
Schaffer Collateral - CA1 Synapse
Postsynaptic Density Membrane
Glutamatergic Synapse
Molecular Function
G-protein Alpha-subunit Binding
G Protein-coupled Receptor Activity
Beta-endorphin Receptor Activity
Voltage-gated Calcium Channel Activity
Protein Binding
Protein C-terminus Binding
Protein Domain Specific Binding
Filamin Binding
G-protein Beta-subunit Binding
Morphine Receptor Activity
Peptide Binding
Neuropeptide Binding
Adenylate Cyclase Inhibiting G Protein-coupled Glutamate Receptor Activity
G Protein-coupled Receptor Activity
Protein Binding
Glutamate Receptor Activity
G Protein-coupled Neurotransmitter Receptor Activity Involved In Regulation Of Postsynaptic Cytosolic Calcium Ion Concentration
G Protein-coupled Receptor Activity Involved In Regulation Of Postsynaptic Membrane Potential
Neurotransmitter Receptor Activity Involved In Regulation Of Postsynaptic Cytosolic Calcium Ion Concentration
Biological Process
Acute Inflammatory Response To Antigenic Stimulus
G Protein-coupled Receptor Signaling Pathway
G Protein-coupled Receptor Signaling Pathway, Coupled To Cyclic Nucleotide Second Messenger
Adenylate Cyclase-inhibiting G Protein-coupled Acetylcholine Receptor Signaling Pathway
Phospholipase C-activating G Protein-coupled Receptor Signaling Pathway
Neuropeptide Signaling Pathway
Sensory Perception
Negative Regulation Of Cell Population Proliferation
Response To Radiation
Cytokine-mediated Signaling Pathway
Sensory Perception Of Pain
Adenylate Cyclase-inhibiting Opioid Receptor Signaling Pathway
Response To Food
Positive Regulation Of Appetite
Response To Lipopolysaccharide
Opioid Receptor Signaling Pathway
Wound Healing
Response To Cocaine
Eating Behavior
Estrous Cycle
Behavioral Response To Ethanol
Positive Regulation Of Neurogenesis
Regulation Of Sensory Perception Of Pain
Excitatory Postsynaptic Potential
Negative Regulation Of Wnt Protein Secretion
Positive Regulation Of ERK1 And ERK2 Cascade
Calcium Ion Transmembrane Transport
Response To Growth Factor
Cellular Response To Morphine
Regulation Of Cellular Response To Stress
Negative Regulation Of Adenylate Cyclase-activating G Protein-coupled Receptor Signaling Pathway
Regulation Of NMDA Receptor Activity
Activation Of MAPKK Activity
Activation Of MAPK Activity
G Protein-coupled Receptor Signaling Pathway
G Protein-coupled Glutamate Receptor Signaling Pathway
Chemical Synaptic Transmission
Locomotory Behavior
Sensory Perception Of Pain
Positive Regulation Of Cytosolic Calcium Ion Concentration Involved In Phospholipase C-activating G Protein-coupled Signaling Pathway
Regulation Of Sensory Perception Of Pain
Regulation Of Synaptic Transmission, Glutamatergic
Regulation Of Postsynaptic Membrane Potential
Cellular Response To Electrical Stimulus
L-glutamate Import Across Plasma Membrane
Regulation Of Postsynaptic Cytosolic Calcium Ion Concentration
Pathways
Opioid Signalling
G-protein activation
Peptide ligand-binding receptors
G alpha (i) signalling events
Interleukin-4 and Interleukin-13 signaling
MECP2 regulates neuronal receptors and channels
G alpha (q) signalling events
Class C/3 (Metabotropic glutamate/pheromone receptors)
Neurexins and neuroligins
Neurexins and neuroligins
Drugs
Tramadol
Morphine
Codeine
Amitriptyline
Hydromorphone
Methadone
Meperidine
Oxycodone
Levallorphan
Dextromethorphan
Butorphanol
Dextropropoxyphene
Pentazocine
Naltrexone
Sufentanil
Alfentanil
Fentanyl
Loperamide
Nalbuphine
Levorphanol
Remifentanil
Ondansetron
Anileridine
Buprenorphine
Hydrocodone
Diphenoxylate
Naloxone
Oxymorphone
Dezocine
Ketamine
Levacetylmethadol
Aripiprazole
Methadyl acetate
3-Methylthiofentanyl
Dimethylthiambutene
Diamorphine
Ethylmorphine
Etorphine
Carfentanil
Diprenorphine
Dihydromorphine
3-Methylfentanyl
V1003
Epicept NP-1
LI-301
Tapentadol
Nalmefene
Alvimopan
Morphine glucuronide
Ketobemidone
Methylnaltrexone
Naloxegol
Cannabidiol
Trimebutine
Butyrfentanyl
Pholcodine
Eluxadoline
Tianeptine
Opium
Pentoxyverine
Naldemedine
Metenkefalin
Medical Cannabis
Nabiximols
Loxicodegol
Oliceridine
Glutamic acid
(S)-alpha-methyl-4-carboxyphenylglycine
Diseases
GWAS
Adult body size (
32376654
)
Body size at age 10 (
32376654
)
Diastolic blood pressure (
30224653
)
HDL cholesterol levels (
32203549
)
Hypertension (
21347282
)
Lipoprotein (a) levels (
26377243
)
Menstruation quality of life impact (fever) (
29855537
)
Methadone dose in opioid dependence (
28115739
)
Opioid use disorder (
32492095
)
Type 2 diabetes (age of onset) (
28060188
)
Cerebral amyloid deposition (PET imaging) (
26252872
)
Suicide (
31476763
)
Waist circumference (
29212154
)
Interacting Genes
77 interacting genes:
ADAM33
ADD3
ALOX5AP
ATP6V0C
ATP6V0E1
C2CD2L
CALM1
CCDC167
CD302
CLCN7
CLDN10
CLDN22
CLDN8
CLEC12B
CLEC7A
CNIH1
COPS5
CPLX1
CTXN3
CYB561
DNAJB4
DOK4
DOK5
EHHADH
EMP1
EMP3
FLNA
GJA4
GNA15
GNAI1
GNAI2
GNAO1
GPRASP1
GRK3
GRM1
HS6ST1
IFITM3
KCNF1
LAT
LPAR3
LRRC25
MAL
MALL
MAP1LC3A
MAP1LC3C
MFF
NELFA
NSG1
OPRD1
OPRL1
PLD2
PLD3
PMP22
PPL
RPRM
RTP4
SCGB1D1
SEC22A
SERP2
SIAH1
SIAH2
SLC30A2
SLC38A7
SLC39A13
SLC41A1
SLC9A9
SMAGP
TEX264
TM4SF4
TMBIM6
TMEM236
TRARG1
UBC
VAPA
WLS
YIPF3
ZYX
40 interacting genes:
ADORA1
BECN1
CABIN1
CASR
CCND2
CCNE1
CD44
CDK4
CDK6
CDKN2B
CDKN2C
EFNB2
EPB41L2
EPHA2
ERBB2
FGFR4
GAPDH
GPRASP1
GRK2
HOMER1
HOMER2
IGF1R
ITPR1
KAT2A
KDELR2
LATS2
MAP2K5
MYC
NF2
OPRM1
OPTN
PDGFRA
PRKCA
RAF1
RASSF1
STK11
TAMALIN
TERT
TTYH2
TUBB
Entrez ID
4988
2911
HPRD ID
02484
05129
Ensembl ID
ENSG00000112038
ENSG00000152822
Uniprot IDs
B8K2Q5
G8XRH4
G8XRH5
L0E130
P35372
Q13255
Q59HC2
PDB IDs
3KS9
4OR2
Enriched GO Terms of Interacting Partners
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Tagcloud (Intersection)
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